Highly Selective Inhibitors Library

Cat. No. :	CS-L158	(4324 compounds)

Library Contents: PDF | SDF

According to reports, most known kinase inhibitors exert their effects through competitive binding in highly conserved ATP pockets. Although genetic techniques such as RNA interference can inactivate specific genes, most kinases are multi domain proteins, each of which has an independent function. Highly selective inhibitors have higher efficiency than non-selective inhibitors, and the selectivity to the target is at least 100 times higher. Therefore, ensuring the validation of targets with the most selective inhibitors is crucial for a more thorough understanding of the pharmacology of the kinase field. The Highly Selective Inhibitors Library contains 4324 compounds, covering multiple targets and subtypes, such as GPCR protein family, Ion channel, multiple kinases, etc. The Highly Selective Inhibitors Library is an effective tool for screening different phenotypes

Size (Pre-dissolved DMSO or Solid)	Stock	Price
30 μL/well (10 mM solution)	In-stock	Get quote
50 μL/well (10 mM solution)	In-stock	Get quote
100 μL/well (10 mM solution)	In-stock	Get quote
250 μL/well (10 mM solution)	In-stock	Get quote

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Data Sheet
Description & Advantages
Composition
Contents

Formulation:	A collection of 4324 highly selective inhibitors supplied as pre-dissolved Solutions or Solid
Container:	96- or 384-well Plate with Peelable Foil Seal; 96-well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:	-80°C
Shipping:	Blue ice or dry ice